Delineating the role of cooperativity in the design of potent PROTACs for BTK [Biochemistry]

Adelajda Zorba, Chuong Nguyen, Yingrong Xu, Jeremy Starr, Kris Borzilleri, James Smith, Hongyao Zhu, Kathleen A. Farley, Wei; Dong Ding, James Schiemer, Xidong Feng, Jeanne S. Chang, Daniel P. Uccello, Jennifer A. Young, Carmen N. Garcia-Irrizary, Lara Czabaniuk, Brandon Schuff, Robert Oliver, Justin Montgomery, Matthew M. Hayward, Jotham Coe, Jinshan Chen, Mark Niosi, Suman Luthra, Jaymin C. Shah, Ayman El-Kattan, Xiayang Qiu, Graham M. West, Mark C. Noe, Veerabahu Shanmugasundaram, Adam M. Gilbert, Matthew F. Brown, Matthew F. Calabrese
National Academy of Sciences
Published 2018