Search Results - (Author, Cooperation:E. Gouaux)
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1Staff View
Publication Date: 2016-04-07Publisher: Nature Publishing Group (NPG)Print ISSN: 0028-0836Electronic ISSN: 1476-4687Topics: BiologyChemistry and PharmacologyMedicineNatural Sciences in GeneralPhysicsKeywords: Allosteric Regulation/drug effects ; Allosteric Site/drug effects ; Antidepressive Agents/chemistry/metabolism/pharmacology ; Citalopram/chemistry/metabolism/pharmacology ; Crystallography, X-Ray ; Dopamine Plasma Membrane Transport Proteins/chemistry ; Drug Design ; Extracellular Space/metabolism ; Humans ; Immunoglobulin Fab Fragments/immunology ; Intracellular Space/metabolism ; Ions/chemistry/metabolism ; Ligands ; Models, Molecular ; Paroxetine/chemistry/metabolism/pharmacology ; Protein Binding/drug effects ; Protein Conformation/drug effects ; Protein Stability ; Serotonin/metabolism ; Serotonin Plasma Membrane Transport Proteins/*chemistry/immunology/*metabolism ; Structure-Activity RelationshipPublished by: -
2C. H. Lee ; W. Lu ; J. C. Michel ; A. Goehring ; J. Du ; X. Song ; E. Gouaux
Nature Publishing Group (NPG)
Published 2014Staff ViewPublication Date: 2014-07-11Publisher: Nature Publishing Group (NPG)Print ISSN: 0028-0836Electronic ISSN: 1476-4687Topics: BiologyChemistry and PharmacologyMedicineNatural Sciences in GeneralPhysicsKeywords: Animals ; Dizocilpine Maleate/chemistry ; Ion Channels/chemistry ; Ligands ; *Models, Molecular ; Phenols ; Piperidines/chemistry ; Protein Binding ; Protein Structure, Tertiary ; Protein Subunits/chemistry ; Receptors, N-Methyl-D-Aspartate/*chemistry ; Xenopus laevis/*physiologyPublished by: -
3Staff View
Publication Date: 2014-08-22Publisher: Nature Publishing Group (NPG)Print ISSN: 0028-0836Electronic ISSN: 1476-4687Topics: BiologyChemistry and PharmacologyMedicineNatural Sciences in GeneralPhysicsKeywords: Allosteric Regulation/drug effects ; Animals ; Apoproteins/*chemistry/metabolism ; Binding Sites ; Binding, Competitive/drug effects ; Caenorhabditis elegans/*chemistry ; Cell Membrane/metabolism ; Chloride Channels/*chemistry/*metabolism ; Crystallography, X-Ray ; Cysteine Loop Ligand-Gated Ion Channel Receptors/*chemistry/*metabolism ; Drug Partial Agonism ; Glutamic Acid/metabolism ; Ion Channel Gating ; Ivermectin/chemistry/metabolism/pharmacology ; Ligands ; Models, Molecular ; Movement/drug effects ; Phosphatidylcholines/chemistry/metabolism/pharmacology ; Protein Binding ; Protein Multimerization/drug effects ; Protein Structure, Tertiary/drug effects ; Structure-Activity RelationshipPublished by: -
4Staff View
Publication Date: 2011-05-17Publisher: Nature Publishing Group (NPG)Print ISSN: 0028-0836Electronic ISSN: 1476-4687Topics: BiologyChemistry and PharmacologyMedicineNatural Sciences in GeneralPhysicsKeywords: Animals ; *Anions ; Binding Sites ; Caenorhabditis elegans/*metabolism ; Chloride Channels/*chemistry/*metabolism ; Cysteine Loop Ligand-Gated Ion Channel Receptors/*metabolism ; Ions/metabolism ; *Models, Molecular ; Neurotransmitter Agents/metabolism ; Protein Structure, TertiaryPublished by: -
5Staff View
Publication Date: 2012-07-31Publisher: Nature Publishing Group (NPG)Print ISSN: 0028-0836Electronic ISSN: 1476-4687Topics: BiologyChemistry and PharmacologyMedicineNatural Sciences in GeneralPhysicsKeywords: Acid Sensing Ion Channels ; Animals ; Binding Sites ; CHO Cells ; Cations, Monovalent/metabolism ; Cesium/metabolism ; Chickens ; Cricetinae ; Crystallography, X-Ray ; Hydrogen-Ion Concentration ; Ion Channel Gating/*drug effects ; Models, Molecular ; Nerve Tissue Proteins/*chemistry/genetics/*metabolism ; Protein Conformation ; Protein Subunits/chemistry/metabolism ; Sequence Deletion ; Sodium/metabolism/pharmacology ; Sodium Channels/*chemistry/genetics/*metabolism ; Spider Venoms/*chemistry/metabolism/*pharmacology ; Spiders/chemistry ; Substrate Specificity/drug effectsPublished by: -
6Staff View
Publication Date: 2012-01-11Publisher: Nature Publishing Group (NPG)Print ISSN: 0028-0836Electronic ISSN: 1476-4687Topics: BiologyChemistry and PharmacologyMedicineNatural Sciences in GeneralPhysicsKeywords: Animals ; Antibodies, Monoclonal/immunology ; Antibody Specificity/immunology ; Apoproteins/*chemistry/genetics/immunology/metabolism ; Bacterial Proteins/*chemistry/genetics/immunology/metabolism ; Binding Sites ; Crystallography, X-Ray ; Immunoglobulin Fab Fragments/immunology ; Ions/chemistry ; Models, Molecular ; Movement ; Protein Conformation ; Sodium/chemistry/metabolism ; Structure-Activity Relationship ; Substrate SpecificityPublished by: -
7Staff View
Publication Date: 2013-09-17Publisher: Nature Publishing Group (NPG)Print ISSN: 0028-0836Electronic ISSN: 1476-4687Topics: BiologyChemistry and PharmacologyMedicineNatural Sciences in GeneralPhysicsKeywords: Animals ; Antidepressive Agents, Tricyclic/chemistry/metabolism/*pharmacology ; Bacterial Proteins/chemistry ; Binding Sites ; Cholesterol/chemistry/metabolism ; Crystallization ; Crystallography, X-Ray ; Dopamine Plasma Membrane Transport Proteins/*chemistry/metabolism ; Drosophila melanogaster/*chemistry ; Ions/chemistry/metabolism ; Models, Molecular ; Nortriptyline/chemistry/metabolism/*pharmacology ; Protein Conformation ; Protein Stability ; Structure-Activity Relationship ; TemperaturePublished by: -
8L. Chen ; K. L. Durr ; E. Gouaux
American Association for the Advancement of Science (AAAS)
Published 2014Staff ViewPublication Date: 2014-08-12Publisher: American Association for the Advancement of Science (AAAS)Print ISSN: 0036-8075Electronic ISSN: 1095-9203Topics: BiologyChemistry and PharmacologyComputer ScienceMedicineNatural Sciences in GeneralPhysicsKeywords: Animals ; Conotoxins/*chemistry ; Conus Snail ; Crystallography, X-Ray ; *Ion Channel Gating ; Ligands ; Mutation ; Protein Binding ; Protein Structure, Secondary ; Protein Structure, Tertiary ; Rats ; Receptors, AMPA/*agonists/*chemistry/geneticsPublished by: -
9H. Wang ; A. Goehring ; K. H. Wang ; A. Penmatsa ; R. Ressler ; E. Gouaux
Nature Publishing Group (NPG)
Published 2013Staff ViewPublication Date: 2013-10-15Publisher: Nature Publishing Group (NPG)Print ISSN: 0028-0836Electronic ISSN: 1476-4687Topics: BiologyChemistry and PharmacologyMedicineNatural Sciences in GeneralPhysicsKeywords: Antidepressive Agents, Second-Generation/metabolism/*pharmacology ; Antidepressive Agents, Tricyclic/metabolism/*pharmacology ; Bacterial Proteins/antagonists & inhibitors/chemistry/genetics/metabolism ; Binding, Competitive/drug effects ; Biogenic Amines/*metabolism ; Chlorides/metabolism ; Crystallography, X-Ray ; Humans ; Mazindol/metabolism/pharmacology ; Models, Molecular ; Mutation ; Norepinephrine/metabolism ; *Plasma Membrane Neurotransmitter Transport Proteins/antagonists & ; inhibitors/chemistry/genetics/metabolism ; Protein Conformation/drug effects ; Recombinant Fusion Proteins/*chemistry/genetics/metabolism ; Reproducibility of Results ; Serotonin Plasma Membrane Transport Proteins/*chemistry/genetics/*metabolism ; Serotonin Uptake Inhibitors/metabolism/*pharmacology ; Sertraline/metabolism/pharmacology ; Sodium/metabolism ; Structure-Activity RelationshipPublished by: -
10Staff View
Publication Date: 2015-05-15Publisher: Nature Publishing Group (NPG)Print ISSN: 0028-0836Electronic ISSN: 1476-4687Topics: BiologyChemistry and PharmacologyMedicineNatural Sciences in GeneralPhysicsKeywords: Animals ; Antidepressive Agents/chemistry/metabolism ; Binding Sites ; Central Nervous System Stimulants/chemistry/*metabolism ; Chlorides/metabolism ; Cocaine/analogs & derivatives/chemistry/metabolism ; Crystallography, X-Ray ; Dextroamphetamine/chemistry/metabolism ; Dopamine/analogs & derivatives/chemistry/metabolism ; Dopamine Plasma Membrane Transport Proteins/*chemistry/*metabolism ; Drosophila melanogaster/*chemistry ; Ligands ; Methamphetamine/chemistry/metabolism ; Models, Molecular ; Molecular Conformation ; Neurotransmitter Agents/chemistry/*metabolism ; Phenethylamines/metabolism ; Protein Stability ; Sodium/metabolismPublished by: -
11Staff View
Publication Date: 2015-09-08Publisher: Nature Publishing Group (NPG)Print ISSN: 0028-0836Electronic ISSN: 1476-4687Topics: BiologyChemistry and PharmacologyMedicineNatural Sciences in GeneralPhysicsPublished by: -
12Staff View
Publication Date: 2012-04-27Publisher: Nature Publishing Group (NPG)Print ISSN: 0028-0836Electronic ISSN: 1476-4687Topics: BiologyChemistry and PharmacologyMedicineNatural Sciences in GeneralPhysicsKeywords: Adenosine Triphosphate/chemistry/*metabolism ; Amino Acid Motifs ; Animals ; Apoproteins/chemistry/metabolism ; Binding Sites ; Crystallization ; Crystallography, X-Ray ; *Ion Channel Gating ; Models, Molecular ; Receptors, Purinergic P2X4/*chemistry/*metabolism ; Structure-Activity Relationship ; ZebrafishPublished by: