Search Results - (Author, Cooperation:D. H. Arlow)
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1R. O. Dror ; T. J. Mildorf ; D. Hilger ; A. Manglik ; D. W. Borhani ; D. H. Arlow ; A. Philippsen ; N. Villanueva ; Z. Yang ; M. T. Lerch ; W. L. Hubbell ; B. K. Kobilka ; R. K. Sunahara ; D. E. Shaw
American Association for the Advancement of Science (AAAS)
Published 2015Staff ViewPublication Date: 2015-06-20Publisher: American Association for the Advancement of Science (AAAS)Print ISSN: 0036-8075Electronic ISSN: 1095-9203Topics: BiologyChemistry and PharmacologyComputer ScienceMedicineNatural Sciences in GeneralPhysicsKeywords: GTP-Binding Protein alpha Subunits, Gi-Go/*chemistry ; GTP-Binding Protein alpha Subunits, Gs/*chemistry ; Guanine Nucleotide Exchange Factors/*chemistry ; Humans ; Models, Chemical ; Molecular Dynamics Simulation ; Protein Structure, Secondary ; Protein Structure, Tertiary ; Receptors, G-Protein-Coupled/*chemistry ; Signal TransductionPublished by: -
2C. Zhang ; Y. Srinivasan ; D. H. Arlow ; J. J. Fung ; D. Palmer ; Y. Zheng ; H. F. Green ; A. Pandey ; R. O. Dror ; D. E. Shaw ; W. I. Weis ; S. R. Coughlin ; B. K. Kobilka
Nature Publishing Group (NPG)
Published 2012Staff ViewPublication Date: 2012-12-12Publisher: Nature Publishing Group (NPG)Print ISSN: 0028-0836Electronic ISSN: 1476-4687Topics: BiologyChemistry and PharmacologyMedicineNatural Sciences in GeneralPhysicsKeywords: Amino Acid Motifs ; Binding Sites ; Crystallization ; Crystallography, X-Ray ; Enzyme Activation/genetics ; Humans ; Hydrolysis ; Lactones/chemistry/pharmacology ; Ligands ; Models, Molecular ; Molecular Dynamics Simulation ; Myocardial Infarction/prevention & control ; Protein Conformation ; Pyridines/chemistry/pharmacology ; Receptor, PAR-1/agonists/antagonists & inhibitors/*chemistry/metabolism ; Receptors, G-Protein-Coupled/chemistry/classification ; Receptors, ThrombinPublished by: -
3R. O. Dror ; H. F. Green ; C. Valant ; D. W. Borhani ; J. R. Valcourt ; A. C. Pan ; D. H. Arlow ; M. Canals ; J. R. Lane ; R. Rahmani ; J. B. Baell ; P. M. Sexton ; A. Christopoulos ; D. E. Shaw
Nature Publishing Group (NPG)
Published 2013Staff ViewPublication Date: 2013-10-15Publisher: Nature Publishing Group (NPG)Print ISSN: 0028-0836Electronic ISSN: 1476-4687Topics: BiologyChemistry and PharmacologyMedicineNatural Sciences in GeneralPhysicsKeywords: Allosteric Regulation/physiology ; Animals ; Binding Sites ; CHO Cells ; Cricetulus ; *Drug Design ; Humans ; Models, Chemical ; Molecular Conformation ; Molecular Dynamics Simulation ; Mutation ; Protein Binding ; Receptors, G-Protein-Coupled/*antagonists & inhibitors/*chemistry/genetics ; Reproducibility of ResultsPublished by: -
4D. M. Rosenbaum ; C. Zhang ; J. A. Lyons ; R. Holl ; D. Aragao ; D. H. Arlow ; S. G. Rasmussen ; H. J. Choi ; B. T. Devree ; R. K. Sunahara ; P. S. Chae ; S. H. Gellman ; R. O. Dror ; D. E. Shaw ; W. I. Weis ; M. Caffrey ; P. Gmeiner ; B. K. Kobilka
Nature Publishing Group (NPG)
Published 2011Staff ViewPublication Date: 2011-01-14Publisher: Nature Publishing Group (NPG)Print ISSN: 0028-0836Electronic ISSN: 1476-4687Topics: BiologyChemistry and PharmacologyMedicineNatural Sciences in GeneralPhysicsKeywords: Adrenergic beta-2 Receptor Agonists/*chemistry/*metabolism ; Crystallization ; Crystallography, X-Ray ; Disulfides/chemistry/metabolism ; Drug Inverse Agonism ; Heterotrimeric GTP-Binding Proteins/metabolism ; Humans ; Lipid Bilayers/chemistry/metabolism ; Models, Molecular ; Molecular Dynamics Simulation ; Procaterol/chemistry/metabolism ; Propanolamines/chemistry/metabolism ; Protein Conformation ; Receptors, Adrenergic, beta-2/*chemistry/*metabolism ; Recombinant Fusion Proteins/chemistry/metabolism ; Viral Proteins/chemistry/metabolismPublished by: -
5A. C. Kruse ; J. Hu ; A. C. Pan ; D. H. Arlow ; D. M. Rosenbaum ; E. Rosemond ; H. F. Green ; T. Liu ; P. S. Chae ; R. O. Dror ; D. E. Shaw ; W. I. Weis ; J. Wess ; B. K. Kobilka
Nature Publishing Group (NPG)
Published 2012Staff ViewPublication Date: 2012-02-24Publisher: Nature Publishing Group (NPG)Print ISSN: 0028-0836Electronic ISSN: 1476-4687Topics: BiologyChemistry and PharmacologyMedicineNatural Sciences in GeneralPhysicsKeywords: Acetylcholine/chemistry/metabolism ; Allosteric Site ; Animals ; COS Cells ; Crystallization ; Crystallography, X-Ray ; Kinetics ; Ligands ; Models, Molecular ; Molecular Dynamics Simulation ; Radioligand Assay ; Rats ; Receptor, Muscarinic M3/*chemistry/*metabolism ; Scopolamine Derivatives/chemistry/metabolism ; Substrate Specificity ; Tiotropium BromidePublished by: